Found 254 from University of Hamburg TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Binding affinity tested against acetylcholinesterase in Torpedo californicaMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 5.30nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity tested against acetylcholinesterase in Torpedo californicaMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Compound tested for inhibition of alpha-galactosidase from Aspergillus nigerMore data for this Ligand-Target Pair
TargetHisto-blood group ABO system transferase(Homo sapiens (Human))
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 1.17E+5nMAssay Description:Inhibition of human blood group B Galactosyltransferase using UDP-Gal as substrate by STD NMR analysis in presence of magnesium ionsMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+5nMAssay Description:Compound tested for inhibition of alpha-galactosidase from Aspergillus nigerMore data for this Ligand-Target Pair
TargetHisto-blood group ABO system transferase(Homo sapiens (Human))
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 3.61E+5nMAssay Description:Inhibition of human blood group B Galactosyltransferase using UDP-Gal as substrate by STD NMR analysis in presence of magnesium ionsMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+5nMAssay Description:Compound tested for inhibition of alpha-galactosidase from Aspergillus nigerMore data for this Ligand-Target Pair
TargetHisto-blood group ABO system transferase(Homo sapiens (Human))
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 5.65E+5nMAssay Description:Competitive inhibition of human blood group B Galactosyltransferase using UDP-Gal as substrate by Michaelis-Menten equation analysis in presence of m...More data for this Ligand-Target Pair
TargetHisto-blood group ABO system transferase(Homo sapiens (Human))
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 5.71E+5nMAssay Description:Inhibition of human blood group B Galactosyltransferase using UDP-Gal as substrate by STD NMR analysis in presence of magnesium ionsMore data for this Ligand-Target Pair
TargetHisto-blood group ABO system transferase(Homo sapiens (Human))
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 1.50E+6nMAssay Description:Inhibition of human blood group B Galactosyltransferase using radiolabeled UDP-Gal as substrate in presence of manganese ionsMore data for this Ligand-Target Pair
TargetHisto-blood group ABO system transferase(Homo sapiens (Human))
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 1.50E+6nMAssay Description:Inhibition of human blood group B Galactosyltransferase using radiolabeled UDP-Gal as substrate in presence of manganese ionsMore data for this Ligand-Target Pair
TargetHisto-blood group ABO system transferase(Homo sapiens (Human))
University Of Hamburg
Curated by ChEMBL
University Of Hamburg
Curated by ChEMBL
Affinity DataKi: 2.20E+6nMAssay Description:Inhibition of human blood group B Galactosyltransferase using radiolabeled UDP-Gal as substrate in presence of manganese ionsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of human MMP13 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human MMP13 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of bovine COX1 assessed as inhibition of calcium ionophore A23187-induced 12-hydroxyheptadecatrienoic acid formation by reverse-phase HPLC...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human MMP9 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human MMP13 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human MMP13 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of human MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of human MMP13 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of human MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Inhibition of human MMP13 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 108nMAssay Description:Inhibition of human MMP9 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of human MMP9 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of COX2 in human whole blood assessed as inhibition of LPS-induced PGE2 synthesis up to 24 hrs by radioimmuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of bovine COX1 assessed as inhibition of calcium ionophore A23187-induced 12-hydroxyheptadecatrienoic acid formation by reverse-phase HPLC...More data for this Ligand-Target Pair
Affinity DataIC50: 151nMAssay Description:Inhibition of human MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 172nMAssay Description:Inhibition of human MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 198nMAssay Description:Inhibition of human MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory activity towards human butyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibitory activity towards human butyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of human MMP13 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 282nMAssay Description:Inhibition of human MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibitory activity towards human butyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of human serum BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibitory activity towards human butyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of bovine COX1 assessed as inhibition of calcium ionophore A23187-induced 12-hydroxyheptadecatrienoic acid formation by reverse-phase HPLC...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of COX2 in human whole blood assessed as inhibition of LPS-induced PGE2 synthesis up to 24 hrs by radioimmuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 503nMAssay Description:Inhibition of human MMP2 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 as substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of bovine 5-LOX assessed as inhibition of calcium ionophore A23187-induced leukotrine B4 formation by reversed phase HPLC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibitory activity towards human butyrylcholinesteraseMore data for this Ligand-Target Pair
